Kiron Canon · Genius, Live Long and Prosper
Peptide Desk
Educational index. Dated 2026-10-27. 152 names.
Caution. This page is educational intelligence. It is not medical advice, not a prescription, and not an offer to sell any compound. BROK does not dose, source, or recommend peptides. Consult a licensed clinician. Athletes must read the current WADA list.
The author's own peptide experimentation is limited because of those risks. Genius, Live Long and Prosper holds that quality protein and collagen ingestion — eggs and collagen supplementation — provide the amino-acid precursor levels a healthy human needs. That is the house first path. Injectables are a specialist medical decision.
Public 152-name map and locators taken from Superpower Health's Peptide Library sitemap and index as of 2026-10-27 (https://x.com/superpower/status/2114785602592035166; https://superpower.com/guides/peptides/). Superpower terms forbid robot copy of their prose; this desk does not rehost their guides. FDA bucket, compounding, WADA, and expanded cards are Nabu classifications from FDA, DailyMed, PubMed, and WADA primary pages. Where a fact is not shown on a primary page, the field says so.
Humans stay free here. Machines: unpaid JSON /peptides.json. Dated claims 50 $POCK or $0.05 USDC at /api/x402/peptides. dest-payTo is in the shop.
71 approved · 26 trials · 34 not approved · 17 cosmetic · 4 withdrawn
FDA-approved (71)
Abaloparatide
Bones & musclesAbaloparatide is an FDA-approved peptide drug. Sold as Tymlos. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Afamelanotide
Skin & agingAfamelanotide is an FDA-approved peptide drug. Sold as Scenesse. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Angiotensin II
Heart & bloodAngiotensin II is an FDA-approved peptide drug. Sold as Giapreza. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Bacitracin
Skin & agingBacitracin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Bivalirudin
Heart & bloodBivalirudin is an FDA-approved peptide drug. Sold as Angiomax. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Bremelanotide
Brain & sleepBremelanotide is an FDA-approved peptide drug. Sold as Vyleesi. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Class. Melanocortin agonist (PT-141 as the research name)
Human evidence. FDA-approved as Vyleesi for acquired, generalized hypoactive sexual desire disorder in premenopausal women. Labelled GI and blood-pressure effects. Not a tanning peptide.
FDA. Approved finished drug. Gray-market PT-141 vials are not that product.
Sport. Approved therapeutic; sport-specific review.
Calcitonin (salmon)
Bones & musclesCalcitonin (salmon) is an FDA-approved peptide drug. Sold as Miacalcin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Cetrorelix
Sexual & reproductiveCetrorelix is an FDA-approved peptide drug. Sold as Cetrotide. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Corticotropin
Hormones & metabolismCorticotropin is an FDA-approved peptide drug. Sold as Acthar. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Cosyntropin
Hormones & metabolismCosyntropin is an FDA-approved peptide drug. Sold as Cortrosyn. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Cyclosporine
Immune & defenseCyclosporine is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Dalbavancin / oritavancin / telavancin
Skin & agingDalbavancin / oritavancin / telavancin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Daptomycin
Skin & agingDaptomycin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Dasiglucagon
Digestive & weightDasiglucagon is an FDA-approved peptide drug. Sold as Zegalogue. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Degarelix
Sexual & reproductiveDegarelix is an FDA-approved peptide drug. Sold as Firmagon. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Desmopressin
Heart & bloodDesmopressin is an FDA-approved peptide drug. Sold as DDAVP. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Difelikefalin
Skin & agingDifelikefalin is an FDA-approved peptide drug. Sold as Korsuva. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Dulaglutide
Hormones & metabolismDulaglutide is an FDA-approved peptide drug. Sold as Trulicity. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Ecallantide
Skin & agingEcallantide is an FDA-approved peptide drug. Sold as Kalbitor. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Echinocandins
Heart & bloodEchinocandins is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Enfuvirtide
Immune & defenseEnfuvirtide is an FDA-approved peptide drug. Sold as Fuzeon. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Eptifibatide
Heart & bloodEptifibatide is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Etelcalcetide
Bones & musclesEtelcalcetide is an FDA-approved peptide drug. Sold as Parsabiv. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Exenatide
Hormones & metabolismExenatide is an FDA-approved peptide drug. Sold as Byetta / Bydureon. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Ga-68 dotatate
Digestive & weightGa-68 dotatate is an FDA-approved peptide drug. Sold as Netspot. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Ganirelix
Sexual & reproductiveGanirelix is an FDA-approved peptide drug. Sold as Ganirelix. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Glucagon
Digestive & weightGlucagon is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Goserelin
Sexual & reproductiveGoserelin is an FDA-approved peptide drug. Sold as Zoladex. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Histrelin
Sexual & reproductiveHistrelin is an FDA-approved peptide drug. Sold as Vantas / Supprelin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Human chorionic gonadotropin
Sexual & reproductiveHuman chorionic gonadotropin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Icatibant
Skin & agingIcatibant is an FDA-approved peptide drug. Sold as Firazyr. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Insulin analogs
Hormones & metabolismInsulin analogs is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Lanreotide
Digestive & weightLanreotide is an FDA-approved peptide drug. Sold as Somatuline. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Leuprolide
Sexual & reproductiveLeuprolide is an FDA-approved peptide drug. Sold as Lupron. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Linaclotide
Digestive & weightLinaclotide is an FDA-approved peptide drug. Sold as Linzess. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Liraglutide
Digestive & weightLiraglutide is an FDA-approved peptide drug. Sold as Victoza / Saxenda. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Lixisenatide
Hormones & metabolismLixisenatide is an FDA-approved peptide drug. Sold as Adlyxin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Lutetium Lu-177 dotatate
Digestive & weightLutetium Lu-177 dotatate is an FDA-approved peptide drug. Sold as Lutathera. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Lutetium Lu-177 vipivotide tetraxetan
Sexual & reproductiveLutetium Lu-177 vipivotide tetraxetan is an FDA-approved peptide drug. Sold as Pluvicto. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Mecasermin
Hormones & metabolismMecasermin is an FDA-approved peptide drug. Sold as Increlex. Desk is educational; a clinician decides use.
WADA S2 · compounding n/a finished drug · public locator
Motixafortide
Heart & bloodMotixafortide is an FDA-approved peptide drug. Sold as Aphexda. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Nafarelin
Sexual & reproductiveNafarelin is an FDA-approved peptide drug. Sold as Synarel. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Octreotide
Digestive & weightOctreotide is an FDA-approved peptide drug. Sold as Sandostatin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Oxytocin
Sexual & reproductiveOxytocin is an FDA-approved peptide drug. Sold as Pitocin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Palopegteriparatide
Bones & musclesPalopegteriparatide is an FDA-approved peptide drug. Sold as Yorvipath. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Parathyroid hormone
Bones & musclesParathyroid hormone is an FDA-approved peptide drug. Sold as Natpara. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Pasireotide
Hormones & metabolismPasireotide is an FDA-approved peptide drug. Sold as Signifor. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Pegcetacoplan
Heart & bloodPegcetacoplan is an FDA-approved peptide drug. Sold as Empaveli / Syfovre. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Pegvisomant
Hormones & metabolismPegvisomant is an FDA-approved peptide drug. Sold as Somavert. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Plecanatide
Digestive & weightPlecanatide is an FDA-approved peptide drug. Sold as Trulance. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Polymyxin B / colistin
Immune & defensePolymyxin B / colistin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Pramlintide
Hormones & metabolismPramlintide is an FDA-approved peptide drug. Sold as Symlin. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
PT-141
Brain & sleepPT-141 is an FDA-approved peptide drug. Sold as research name of bremelanotide (Vyleesi). Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Secretin
Hormones & metabolismSecretin is an FDA-approved peptide drug. Sold as ChiRhoStim. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Semaglutide
Digestive & weightSemaglutide is an FDA-approved peptide drug. Sold as Ozempic / Wegovy / Rybelsus. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Class. GLP-1 receptor agonist
Human evidence. STEP 1 (NEJM): ~14.9% mean weight loss vs 2.4% placebo at 68 weeks. SELECT (NEJM): 20% reduction in major cardiovascular events (HR 0.80) in 17,604 adults with overweight/obesity and established CVD without diabetes.
FDA. FDA-approved as Ozempic, Wegovy, and Rybelsus for labelled uses including type 2 diabetes, chronic weight management, cardiovascular risk reduction, CKD in T2D, and noncirrhotic MASH (Wegovy). Boxed warning for thyroid C-cell tumors in rodents.
Sport. Approved therapeutic; athletes still need sport-specific review.
Setmelanotide
Digestive & weightSetmelanotide is an FDA-approved peptide drug. Sold as Imcivree. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Sincalide
Digestive & weightSincalide is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Somapacitan
Hormones & metabolismSomapacitan is an FDA-approved peptide drug. Sold as Sogroya. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Somatropin (rhGH)
Hormones & metabolismSomatropin (rhGH) is an FDA-approved peptide drug. Sold as Genotropin and others. Desk is educational; a clinician decides use.
WADA S2 · compounding n/a finished drug · public locator
Teduglutide
Digestive & weightTeduglutide is an FDA-approved peptide drug. Sold as Gattex. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Teriparatide
Bones & musclesTeriparatide is an FDA-approved peptide drug. Sold as Forteo. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Terlipressin
Digestive & weightTerlipressin is an FDA-approved peptide drug. Sold as Terlivaz. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Tesamorelin
Digestive & weightTesamorelin is an FDA-approved peptide drug. Sold as Egrifta. Desk is educational; a clinician decides use.
WADA S2 · compounding n/a finished drug · public locator
Class. GHRH analogue
Human evidence. Approved as Egrifta for reduction of excess abdominal fat in HIV-associated lipodystrophy. Off-label and compounded versions are a different legal object.
FDA. FDA-approved branded product. Compounded/off-label tesamorelin is a separate row on this desk.
Sport. S2 peptide hormone analogue in sport.
- P1 · DailyMed tesamorelin
- P1 · WADA Prohibited List
Tirzepatide
Digestive & weightTirzepatide is an FDA-approved peptide drug. Sold as Mounjaro / Zepbound. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Class. GIP/GLP-1 receptor agonist
Human evidence. SURMOUNT-1 reported ~20.9% mean weight loss at 15 mg over 72 weeks in a separate trial from STEP 1. Dual-incretin, not interchangeable with semaglutide.
FDA. FDA-approved as Mounjaro (T2D) and Zepbound (weight). Labelled drug; clinician-prescribed.
Sport. Approved therapeutic; sport-specific review.
Triptorelin
Sexual & reproductiveTriptorelin is an FDA-approved peptide drug. Sold as Trelstar. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Trofinetide
Brain & sleepTrofinetide is an FDA-approved peptide drug. Sold as Daybue. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Vancomycin
Heart & bloodVancomycin is an FDA-approved peptide drug. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Vasopressin
Heart & bloodVasopressin is an FDA-approved peptide drug. Sold as Vasostrict. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Vosoritide
Bones & musclesVosoritide is an FDA-approved peptide drug. Sold as Voxzogo. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Ziconotide
Brain & sleepZiconotide is an FDA-approved peptide drug. Sold as Prialt. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
Zilucoplan
Bones & musclesZilucoplan is an FDA-approved peptide drug. Sold as Zilbrysq. Desk is educational; a clinician decides use.
WADA therapeutic_check_list · compounding n/a finished drug · public locator
US product withdrawn / discontinued (4)
Albiglutide
Hormones & metabolismAlbiglutide was FDA-approved and later left the US market. Sold as Tanzeum (withdrawn).
WADA unknown_verify · compounding n/a finished drug · public locator
Desirudin
Heart & bloodDesirudin was FDA-approved and later left the US market. Sold as Iprivask (discontinued).
WADA unknown_verify · compounding n/a finished drug · public locator
Nesiritide
Heart & bloodNesiritide was FDA-approved and later left the US market. Sold as Natrecor (discontinued).
WADA unknown_verify · compounding n/a finished drug · public locator
Sermorelin
Bones & musclesSermorelin was FDA-approved and later left the US market. Sold as Geref (discontinued).
WADA S2 · compounding n/a finished drug · public locator
Class. GHRH 1-29 analogue
Human evidence. Geref was FDA-approved then discontinued. Compounded sermorelin is not the discontinued branded product.
FDA. Finished US product discontinued. Compounded copies are a separate legal question.
Sport. S2.
- P1 · WADA
In clinical trials (26)
Amycretin
Digestive & weightAmycretin is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Apraglutide
Digestive & weightApraglutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Aviptadil
Immune & defenseAviptadil is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Balixafortide
Heart & bloodBalixafortide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Brilacidin
Digestive & weightBrilacidin is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Cagrilintide
Digestive & weightCagrilintide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
CagriSema
Digestive & weightCagriSema is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Davunetide
Brain & sleepDavunetide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Efpeglenatide
Hormones & metabolismEfpeglenatide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Elamipretide
Hormones & metabolismElamipretide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Enlicitide
Digestive & weightEnlicitide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Glepaglutide
Digestive & weightGlepaglutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Larazotide acetate
Digestive & weightLarazotide acetate is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
LTX-315
Skin & agingLTX-315 is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Mazdutide
Digestive & weightMazdutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Murepavadin
Immune & defenseMurepavadin is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Nangibotide
Immune & defenseNangibotide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
NNZ-2591
Brain & sleepNNZ-2591 is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Pemvidutide
Digestive & weightPemvidutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Petrelintide
Digestive & weightPetrelintide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
PN-943
Digestive & weightPN-943 is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Retatrutide
Digestive & weightRetatrutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Rusfertide
Heart & bloodRusfertide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Selepressin
Heart & bloodSelepressin is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Survodutide
Digestive & weightSurvodutide is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Trofinetide predecessor programs
Brain & sleepTrofinetide predecessor programs is in clinical development. Not an approved US drug as of 2026-10-27.
WADA unknown_verify · compounding closed or unlisted · public locator
Not FDA-approved (34)
5-Amino-1MQ
Digestive & weightsmall molecule5-Amino-1MQ is a small molecule often sold next to peptides. FDA compounding risk listed. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
AOD-9604
Digestive & weightAOD-9604 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding nominated withdrawn · public locator
Class. HGH fragment analogue
Human evidence. FDA withdrawn-nomination page: immunogenicity / impurity; limited safety information; serious adverse events mentioned with causality unclear.
FDA. Not approved.
Sport. S0 typical.
- P1 · FDA compounding page
BPC-157
Digestive & weightBPC-157 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding nominated withdrawn · public locator
Class. Synthetic pentadecapeptide (gastric-derived fragment)
Human evidence. HSS Journal 2025 systematic review: 36 studies included, 35 preclinical, 1 retrospective human series n=12 with no control and no safety table (PMID 40756949).
FDA. Never FDA-approved. Nominated for 503A compounding then withdrawn April 2026. Still not on the 503A bulks list or Category 1. PCAC July 2026 vote is advisory. Licensed US compounding remains closed as of this desk date.
Sport. WADA S0 Non-Approved Substances. Prohibited at all times in sport.
Cerebrolysin
Brain & sleepCerebrolysin is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
CJC-1295
Bones & musclesCJC-1295 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding nominated withdrawn · public locator
Class. GHRH analogue (with or without DAC)
Human evidence. FDA lists CJC-1295 under nominated-but-withdrawn compounding substances with heart-rate and vasodilatory adverse-event language. Available clinical data are limited.
FDA. Nominated then withdrawn from Category 2. Still not a cleared 503A bulk.
Sport. S2.
- P1 · FDA compounding page
- P1 · WADA
Gonadorelin (compounded)
Sexual & reproductiveGonadorelin (compounded) is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding closed or unlisted · public locator
Tesamorelin (off-label / compounded)
Hormones & metabolismTesamorelin (off-label / compounded) is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
Dihexa
Brain & sleepDihexa is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
DSIP (emideltide)
Brain & sleepDSIP (emideltide) is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding nominated withdrawn · public locator
Epitalon
Brain & sleepEpitalon is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding nominated withdrawn · public locator
Class. Synthetic tetrapeptide (Ala-Glu-Asp-Gly)
Human evidence. FDA: nominated-but-withdrawn; immunogenicity / aggregation language; no adequate human safety package on the compounding page.
FDA. Not approved. Compounding closed.
Sport. S0 typical for non-approved substances.
- P1 · FDA compounding page
Follistatin-344
Bones & musclesFollistatin-344 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
HGH fragment 176-191
Digestive & weightHGH fragment 176-191 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
GHK-Cu
Skin & agingGHK-Cu is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding nominated withdrawn · public locator
Class. Copper tripeptide
Human evidence. Topical cosmetic use is common. FDA lists injectable GHK-Cu under nominated-but-withdrawn compounding with immunogenicity language and limited human data.
FDA. Injectable compounding closed. Topical cosmetic is a different object.
Sport. Typical none for topical cosmetic; verify if injected.
- P1 · FDA compounding page
GHRP-2
Bones & musclesGHRP-2 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding category 2 · public locator
Class. Growth-hormone releasing peptide
Human evidence. FDA Category 2 (503B) for injectable and nasal routes: immunogenicity, unnatural amino acid, reports of serious events with causality not established.
FDA. Category 2. Not approved.
Sport. S2.
- P1 · FDA Category 2 page
GHRP-6
Bones & musclesGHRP-6 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding category 2 · public locator
Class. Growth-hormone releasing peptide
Human evidence. FDA Category 2 (503B): immunogenicity / impurity language; cortisol and glucose effects in available data.
FDA. Category 2. Not approved.
Sport. S2.
- P1 · FDA Category 2 page
Hexarelin
Bones & musclesHexarelin is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
Humanin
Hormones & metabolismHumanin is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
IGF-1 DES
Bones & musclesIGF-1 DES is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
IGF-1 LR3
Bones & musclesIGF-1 LR3 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
Ipamorelin
Bones & musclesIpamorelin is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding category 2 · public locator
Class. Ghrelin-mimetic GHRP
Human evidence. No FDA-approved finished drug. FDA Category 2 under 503B for ipamorelin acetate (immunogenicity / impurity / IV motility study deaths in literature; causality not always established).
FDA. Category 2 on FDA compounding safety page as of this desk date. Not a 503A bulk.
Sport. S2 peptide hormones and growth-factor mimetics.
Kisspeptin-10
Sexual & reproductiveKisspeptin-10 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding category 2 · public locator
Class. Kisspeptin fragment
Human evidence. FDA Category 2 (503A): immunogenicity / impurity; limited safety information for proposed routes.
FDA. Category 2. Not approved as a finished US drug.
Sport. Verify current WADA list.
- P1 · FDA Category 2 page
KPV
Digestive & weightKPV is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding nominated withdrawn · public locator
LL-37 (cathelicidin)
Immune & defenseLL-37 (cathelicidin) is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding nominated withdrawn · public locator
Class. Human cathelicidin antimicrobial peptide
Human evidence. FDA withdrawn-nomination page: limited human safety; nonclinical notes include male-reproduction and protumorigenic signals in some tissues.
FDA. Not approved. Nominated then withdrawn.
Sport. Verify list.
- P1 · FDA compounding page
Mechano growth factor
Bones & musclesMechano growth factor is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding nominated withdrawn · public locator
Melanotan I
Skin & agingMelanotan I is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding closed or unlisted · public locator
Melanotan II
Skin & agingMelanotan II is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding nominated withdrawn · public locator
Class. Melanocortin agonist
Human evidence. Not FDA-approved. FDA compounding page lists immunogenicity / impurity language. Case reports of priapism and pigment change circulate in the literature.
FDA. Nominated-but-withdrawn compounding substance. Unapproved.
Sport. Verify current WADA list; often treated as prohibited.
- P1 · FDA compounding page
MK-677 (ibutamoren)
Bones & musclessmall moleculeMK-677 (ibutamoren) is a small molecule often sold next to peptides. FDA compounding risk listed. Educational desk only.
WADA S4 · compounding category 2 · public locator
Class. Non-peptide ghrelin-receptor agonist (small molecule)
Human evidence. FDA Category 2: a hip-fracture recovery RCT was terminated early for a congestive-heart-failure safety signal.
FDA. Category 2 for 503A and 503B. Not an approved drug. Not a peptide.
Sport. S4 hormone and metabolic modulators (ibutamoren).
- P1 · FDA Category 2 page
- P1 · WADA
MOTS-c
Hormones & metabolismMOTS-c is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
Class. Mitochondrial-derived peptide
Human evidence. No FDA-approved product. Human evidence remains early.
FDA. Not approved. Superpower states it does not facilitate research-only MOTS-c.
Sport. Treat as non-approved / verify list.
- P1 · WADA Prohibited List
Selank
Brain & sleepSelank is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
Semax
Brain & sleepSemax is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
TB-500
Bones & musclesTB-500 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
Class. Synthetic fragment of thymosin beta-4
Human evidence. No completed controlled human efficacy trials as an FDA-approved drug. Often discussed with BPC-157 in recovery forums; different sequence and mechanism.
FDA. Not FDA-approved.
Sport. S2 (thymosin beta-4 / related fragments).
- P1 · WADA Prohibited List
Thymosin alpha-1
Immune & defenseThymosin alpha-1 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA unknown_verify · compounding closed or unlisted · public locator
Thymosin beta-4
Bones & musclesThymosin beta-4 is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S2 · compounding closed or unlisted · public locator
Thymulin
Immune & defenseThymulin is not FDA-approved for any human use. Human evidence is thin or absent. Educational desk only.
WADA S0 · compounding closed or unlisted · public locator
Cosmetic / topical (17)
Acetyl hexapeptide-8
Skin & agingAcetyl hexapeptide-8 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Acetyl octapeptide-3
Skin & agingAcetyl octapeptide-3 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Acetyl tetrapeptide-5
Skin & agingAcetyl tetrapeptide-5 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Carnosine
Skin & agingCarnosine is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Copper tripeptide-1
Skin & agingCopper tripeptide-1 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Dipeptide diaminobutyroyl benzylamide diacetate
Skin & agingDipeptide diaminobutyroyl benzylamide diacetate is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Glutathione
Skin & agingGlutathione is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Hexapeptide-9
Skin & agingHexapeptide-9 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Nonapeptide-1
Skin & agingNonapeptide-1 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Oligopeptide-1
Skin & agingOligopeptide-1 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Palmitoyl hexapeptide-12
Skin & agingPalmitoyl hexapeptide-12 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Palmitoyl pentapeptide-4
Skin & agingPalmitoyl pentapeptide-4 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Palmitoyl tetrapeptide-7
Skin & agingPalmitoyl tetrapeptide-7 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Palmitoyl tripeptide-1
Skin & agingPalmitoyl tripeptide-1 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Palmitoyl tripeptide-38
Skin & agingPalmitoyl tripeptide-38 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Pentapeptide-18
Skin & agingPentapeptide-18 is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Tripeptide-10 citrulline
Skin & agingTripeptide-10 citrulline is used in topical cosmetic formulas. Not an FDA-approved injectable drug.
WADA none_typical · compounding n/a cosmetic · public locator
Desk date 2026-10-27. Re-open FDA before any compounding sentence. Not financial, legal, or medical advice.